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Active Pharmaceuticals

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Product nomen: Magnesium esomeprazole
Originale China
CAS 161973-10-0
Formulae hypotheticae C34H36MgN6O6S2
M. Pondus 713.12

Esomeprazole venditum notam nomine Nexium apud alios, Est protón-sentinam inhibitor quae reduces stomachum acidum. Ponitur in curatione dyspepsiae, morbus ulceris peptic, refluxus gastroesophageus morbus, et Zollinger-Elison syndrome.

Decrescit secretionem acidi per inhibitionem H+/K+-ATPase in cellulis parietalibus ventriculi. Per hoc transporter inhibentes operationem, medicamentum prohibet formationem stomachi acid.Esomeprazole est (S)-(−)-enantiomer de omeprazole. Esomeprazole is currently sold over the counter in the US and the UK.

Esomeprazole is used to treat certain stomach and esophagus problems (such as acid reflux, ulceribus). It works by decreasing the amount of acid your stomach makes. It relieves symptoms such as heartburn, difficulty swallowing, and persistent cough. This medication helps heal acid damage to the stomach and esophagus, helps prevent ulcers, and may help prevent cancer of the esophagus. Esomeprazole belongs to a class of drugs known as proton pump inhibitors (PPIs).

If you are self-treating with this medication, over-the-counter esomeprazole products are used to treat frequent heartburn (occurring 2 or more days a week). Since it may take 1 to 4 days to have full effect, these products do not relieve heartburn right away.

Primi usus esomeprazolis sunt morbo refluxus gastroesophagi, curatio et sustentationem erosivae gulae, curatio ulcerum duodenalium per H *. pylori, ne ulcera gastrica in his chronicis NSAID, et curationem ulcerum gastrointestinalium cum morbo Crohn adjunctis.

Esomeprazole is available ut moratus-release capsulae in Civitatibus Foederatis Americae, vel ut tabulas in Australia moratus-release, Britanniae, et Canada (magnesium continet esomeprazole) per robora of * 20 et 40 mg, sicut moratus-release capsulae in Civitatibus Foederatis Americae (esomeprazole strontium continet) in a * 49.3 mg vi (equivalent of * delivering 40 emptum esomeprazole, et sicut esomeprazole sodium pro infusione intravenous/infusion. Praeparata esomeprazole orali sunt enterico-coactata, ex celeri deiectione medicamento in acidis conditionibus stomachi. Hoc fit per capsulas formandas utendo systematis multi-unitatis globulo.

Magnesium esomeprazolum etiam cum naproxeno coniungitur (sub notam nomine Vimovo) ad praeventionis ulcera gastrica cum longis NSAID illic consociata. Vimovo is available in 2 dosis vires: 500/20 mg. & 375/20 mg. Tribulationes Pivotal clinicae Vimovo (apud " 6 mensis finem punctum) demonstrandum incidentia GI ulceris in 24% de aegris in naproxen (solus) versus 7% de naproxen/esomeprazole. The FDA admonitiones ad pittacium de Viomovo de nephritis acutis interstitialibus addidit, renibus problems in aliquo aegris periculum.

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