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Antiestrogen Steroids

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CAS: 107868-30-4
Formulae hypotheticae: C20H24O2
M. pondus:296.4
Gradus : Pharmaceutical Grade
Repono: Shading, inclusi conservationem

Exemestane (nomen artis Aromasin) est medicamento ad facies carcinomate. Membrum est genus medicamentorum asaromatarum notarum inhibitores. Quidam carcinomata sua require estrogen crescere. Carcinomata illae receptores estrogen (ERs), et vocantur ER-positive. They may also called estrogen-responsive, hormonally-responsive,aut hormone-receptorpositive.Aromatase est enzyme quod estrogen. Aromatase inhibitors synthesin angustos estrogenium. Hoc gradu estrogen demittit, et incrementum carcinomata sua praepedit.

Exemestane est oralis aromatasi steroidalis inhibitoris quae in ER-positivo cancer pectoris adhibetur praeter chirurgicam et/vel radialem in feminis post-menopausalis. Aromasin pugnare cancer pectus et testosteronem in corpore suscitat. Exemestane processum aromatisationis impedit.. Estrogenium igitur quantitatem demittit in corpore. In primo cancer, exemestane potest auxilium prohibere cancer veniens retro. In cancro carcinomate provecto cellae cancer tardius crescere vel desinere totaliter crescere potest.

Exemestane aromatasi est inhibitor. Id impedit enzyme aromatase (in corporis musculus, pellis, pectus et pinguis), quod adhibetur ut convertat androgens (hormones produci glandulae) in estrogen. In absentia estrogen, tumores ab hoc hormone dependentes ad incrementum recusabunt.

Exemestane portat facultatem inhibendi aromatase enzyme, quae productio vel conversio testosteronis est in estrogen. Aromasin habet facultatem aromatization angustos, quae rursus productio estrogenium vetat, eoque demittit corpus gradus estrogenium.

Test items SPECIFICATION Effectus
Descriptio Crystallina pulveris alba Alba pulveris
Lepidium sativum Positivum Positivum
Assay(per HPLC *) 98.0~102.0% 99.64%
Absorbance(E1cm) 465~495 482.5
Liquefactio Point 191~195℃ 193.5~195.0℃
Damnum de Siccatio 0.5%max 0.19%
Imprimis Rotationes +288°~ +298° +290.2°
Residua de Ignition 0.1%max 0.03%
Substantiae cognatae Totalis:1.5%max <1.3%
Residuum Solvents 0.2%max 0.10%
Metalla gravis 20PPm max <10PPm
conclusio Specificatio conformis USP35

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