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Active Pharmaceuticals

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Product Name:Onapristone

CAS:96346-61-1

MF:C29H39NO3

MW:449.62

Onapristone (INN) (nomina in codice developmental ZK-89299, ZK-299) est synthetica et steroidalis antiprogestogen cum additamento antiglucocorticoidei operationis quae a Schering evoluta est et descripta. 1984 sed numquam fuit (PR), antiprogestogen mifepristone actis contraque (quod est infirmum receptoris partialis agonist).Praeterea, comparari mifepristone, onapristone redegit antiglucocorticoid operatio, parum antiandrogenic activitatem, et habet 10- ad 30-ovili maiorem potentiam ut antiprogestogen. The medication was under development for clinicus usus est, puta in curatione cancri pectoris et ut contraceptivum endometriale, sed discontinuata est durante periodo III in iudiciis clinicis 1995 ob inventa iecoris munus abnormitates quam in pluribus aegris.

Onapristone efficax in curatione carcinomatis repertus est.

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