製品名:Taltirelin Acetate
別名:TA-0910 Acetate;Ceredist
CAS:1549593-23-8
MF:C19H27N7O7
MW:465.47
Taltirelin acetate (TA-0910 アセテート) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Taltirelin Acetate is an analogue of protirelin (Go to Protirelin) and is claimed to have beneficial effects on CNS function. It is used in the treatment of spinocerebellar degeneration.
| 分子式: |
C17H31N7○9 |
| 分子量: |
477.46 |
| CAS番号: |
103300-74-9 |
| 外観: |
白い粉 |
| ペプチド含有量(by %N): |
≥80% |
| アセテート含有量(HPLCによる): |
≤15% |
| 純度(HPLCによる): |
0.98 |
| 単一の不純物(HPLCによる): |
≤1.0% |
| アッセイ(By Anhydrous, Acetic Acid-free): |
95.0～105.0% |
| MS: |
一貫性のある |
