Produk Naam:Taltirelin-asetaat
Ander Naam:TEKEND-0910 Asetaat;Ceredist
CAS:1549593-23-8
MF:C19H27N7O7
MW:465.47
Taltirelin acetate (TEKEND-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Taltirelin Acetate is an analogue of protirelin (Go to Protirelin) and is claimed to have beneficial effects on CNS function. It is used in the treatment of spinocerebellar degeneration.
| Molekulêre Formule: |
C17H31N7O9 |
| Molekulêre gewig: |
477.46 |
| CAS No.: |
103300-74-9 |
| Voorkoms: |
Wit poeier |
| Peptied inhoud(deur %N): |
≥80% |
| Asetaat inhoud(deur HPLC): |
≤15% |
| Reinheid(deur HPLC): |
0.98 |
| Enkele Onreinheid(deur HPLC): |
≤1,0% |
| Assay(Deur Anhydrous, Asynsuurvry): |
95.0~105,0% |
| MS: |
Konsekwent |