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Active Pharmaceuticals

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Product Name: Vinblastine sulfate
Synonyma: 29060le;exal;nsc49842;rozevinsulfate;velban;velbe;vincaleukoblastine,sulfate(1:1)(salt);Vinblastine, sulphate salt
CAS: 143-67-9
MF: C46H60N4O13S
MW: 909.05
EINECS: 205-606-0

Vinblastine is a medication used to treat a number of types of cancer including: Hodgkin's lymphoma, non-small cell lung cancer, bladder cancer, brain cancer, and testicular cancer among others.It is used intravenously and works by inhibiting mitosis.

1. It has vasodilating, blood thinning, and memory-enhancing actions.

2. It acts as a cerebral stimulant and vasodilator.

3. It is used to treat arteriosclerosis.

4. It is very effective in curing dementia caused due to insufficient blood supply to the brain.

5. It interferes with cells' ability to synthesize DNA and RNA.

Mainly used for the treatment of solid tumor. For malignant lymphoma, testicular neoplasm and choriocarcinoma curative effect is better. For lung, pectus, ovarian, skin cancer, renal mother cell tumor and monocytes leukaemia also have certain curative effect.

Items Signa Proventus
Aspectus Alba vel off-alba solidum pulveris Obsequitur
Lepidium sativum per IR Obsequitur
per HPLC Obsequitur
Solubilitas Solutum in DMF *, parce solutum in THF *, slightly soluble in methanol and acetonitrile, very sightly soluble in ethanol and dichloromethane, insolubilem aquam Obsequitur
Forma polymorphica Forma polymorphica 1 Obsequitur
Liquefactio Point 211C~216ºC 212.8C~ 214.9ºC
Aqua Content ≤ 0.50% 0.10%
Metalla gravis ≤ 20ppm Obsequitur
Residere in Ignition ≤ 0.20% 0.09%
Substantia cognata Si una immunditia: ≤0.10% 0.06%
Totalis immunditias: ≤1.00% 0.16%
Assay (in anhydrous basis) 98.0%~102.0% 99.94%
Magnitudo particula D90: ≤100µm Obsequitur
Reference Standard In-domus Latin
conclusio Productum obtemperavit in domo vexillum.

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