Chemiese naam: Asetildenafil
CAS: 831217-01-7
Sinonieme: Hongdenafil;Asetildenafil;Asetildenafil (Hongdenafil);5-[2-Etoksie-5-[2-(4-etiel-piperasien-1-yl)-asetiel]-feniel]-1-Metiel-3-propiel-1,6-dihidro-pirazolo[4,3-d]pyriMidin-7-one;5-[2-Etoksie-5-[2-(4-etiel-1-piperasiniel)asetiel]feniel]-1,6-dihidro-1-metiel-3-propiel-7H-pirazolo[4,3-d]pirimidin-7-een;7H-Pyrazolo[4,3-d]pyriMidin-7-one,
Molekulêre Formule: C25H34N6O3
Formule gewig: 466.583
Assay: 99%
LP: 131-133°C
Berging temp: Yskas
Chemiese Eienskappe: Naaswit tot liggeel solied
Gebruik: Acetildenafil is 'n middel wat gebruik word om erektiele disfunksie te behandel (impotensie) by mans en pulmonale arteriële hipertensie (PAH).
Acetildenafil is 'n sintetiese middel wat bekend is dat dit optree as 'n fosfodiesterase-inhibeerder. Dit is 'n analoog van sildenafil (Viagra) en blykbaar libido 'n hupstoot te gee en erektiele disfunksie te verlig. Sedert, Acetildenafil inhibeer fosfodiesterase-ensiem, dit kan gebruik word om intrasellulêre vlakke van die tweede boodskappers cAMP en cGMP te reguleer, en selfunksie.
Ten spyte van sulke belowende effekte van hierdie stof, Acetildenafil bly 'n navorsingschemikalie, word hoofsaaklik deur navorsers van regoor die wêreld gebruik om wetenskaplike eksperimente uit te voer. Geen deeglike toetsing op die bogenoemde effekte van asetildenafiel is tot dusver uitgevoer nie. Wetenskaplikes kan navorsing doen oor hierdie potensiële chemikalie om meer te wete te kom oor die voordelige gebruike daarvan.
- Dit kan optree as 'n inhibeerder van fosfodiesterase
Asetildenafil kan fosfodiesterase inhibeer 5, wat beteken dit kan die afbrekende werking van cGMP-spesifieke fosfodiesterase tipe blokkeer 5 (PDE5) on cyclic GMP present in the smooth muscle cells of the blood vessels that supply blood to male genital organs. Recently, Acetildenafil has been detected in a number of over-the-counter herbal aphrodisiac products.
- It acts as a Vasodilator Agent
Vasodilator Agents are synthetic drugs used to cause dilation of the blood vessels, therefore cause a decrease in vascular resistance and an increase in blood flow. With further research on the effects of acetildenafil and its analogues on blood vessels, it will enable researchers to understand how it could be beneficial for treating hypertension, wherein the patient has high blood pressure as well as congestive heart failure.
- It acts as a Urological Agent
Urological Agents are drugs used in the treatment of urogenital conditions such as urinary incontinence, erectile dysfunction and prostatic hyperplasia. Acetildenafil acts as urological agent because it inhibits the enzyme - phosphodiesterase type 5 (PDE5). Blocking PDE5 promotes the development and maintenance of male genital stimulation.
| Item |
Requirement |
Resultate |
| Beskrywing |
Wit poeier |
Wit poeier |
| Smeltpunt |
191192 |
192 |
| Red outside |
according to medical standard |
complies |
| Absorption of ultravioletradiation |
290nm massive of absorption |
Konformeer |
| Verlies by droog |
<.5% |
0.30% |
| Swaar metale |
<20dpm |
10dpm |
| assay |
99.00% |
99.90% |
| conclusion |
The product conforms to enterprise standard |
