Product Name:Taltirelin Acetate
Other Name:TA-0910 Acetate;Ceredist
CAS:1549593-23-8
MF:C19H27N7O7
MW:465.47
Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release).
Taltirelin Acetate is an analogue of protirelin (Go to Protirelin) and is claimed to have beneficial effects on CNS function. It is used in the treatment of spinocerebellar degeneration.
| Molecular Formula: |
C17H31N7O9 |
| Molecular Weight: |
477.46 |
| CAS No.: |
103300-74-9 |
| Appearance: |
White powder |
| Peptide Content(by %N): |
≥80% |
| Acetate Content(by HPLC): |
≤15% |
| Purity(by HPLC): |
0.98 |
| Single Impurity(by HPLC): |
≤1.0% |
| Assay(By Anhydrous, Acetic Acid-free): |
95.0~105.0% |
| MS: |
Consistent |
