酢酸カルベトシン
順序: ブチリル-チル(自分)-Ile-Gln-Asn-Cys-Pro-Leu-Gly-NH2 (ブチリル-4-イルとCysの間のスルフィド結合)
CAS: 37025-55-1
外観: 白い粉
アイネス: 253-312-6
MF: C45H69N11O12S
M.W.: 988.17
比旋光度 D(c=1.1% HAc): -38.0~-42.0°
水分含有量(カール・フィッシャー): ≤5.0%
アセテート含有量(HPLCによる): ≤12.0%
アミノ酸組成: 理論値の±10%
純度 (HPLCによる): ≧98.0%
単一の不純物(HPLCによる): ≤1.0%
ペプチド含有量(N%まで): ≥80%
アッセイ(無水で, 酢酸フリー ): 97.0~103.0%
細菌エンドトキシン: ≤5EU/mg
使用法:An obstetric drug used to control postpartum hemorrhaging.
Carbetocin (宿, 禁止) (brand names Duratocin, Pabal, Lonactene, Depotocin, Comoton, Decomoton), or 1-butanoic acid-2-(O-methy-L-tyrosine)-1-carbaoxytocin, is an oxytocic used in obstetrics to control postpartum hemorrhage and bleeding after giving birth, particularly following Cesarean section. It is an eight amino acid long analogue of oxytocin (a nonapeptide) そして, それに応じて, has a similar action. Carbetocin primarily agonizes peripherally expressed oxytocin receptors.
Carbetocin is an oxytocic used in obstetrics to control postpartum hemorrhage and bleeding after giving birth, particularly following Cesarean section. It is an eight amino acid long analogue of oxytocin (a nonapeptide) そして, それに応じて, has a similar action. Carbetocin primarily agonizes peripherally expressed oxytocin receptors.